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Publications + Posters
|
Journal of Biological Chemistry
October 2026
Genetic and biochemical screens identify MGAT1 as a druggable glycosyltransferase target in STK11-mutant lung cancer
Kiera M. Vassallo, et al.
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Discovery on Target
September 2026
Covalent and Non-Covalent Lead Generation Strategies for VRK1, a Paralog Synthetic Lethal Target in Cancer
Kasia Handing
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Gordon Research Conference: Enzymes, Coenzymes and Metabolic Pathways
July 2026
Mass Spectrometry-Based Kinetic and Site-Specific Profiling of Covalent Inhibitors Targeting VRK1
Mu-Sen Liu
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Chemical Computing Group North American User Group Meeting & Conference
June 2026
Hit finding and assay enablement for MGAT1, a novel glycosyltransferase involved in cancer cell immune evasion
Kasia Handing
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AACR Cancer Research
June 2026
TNG917 is a Potent and Selective Inhibitor of Histone Lysine Methyltransferases EHMT1/2 that Enhances Antitumor Immunity and Immunotherapy Efficacy
Alvin Ziying Lu, et al.
Learn more about our drug discovery programs and explore our pipeline.